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Articles

Vol. 2 No. 3 (2011): July – September 2011

Synthesis and antimicrobial activity of 5-aminoquinoline and 3-amino phenol derivatives

DOI
https://doi.org/10.37285/ijddd.2.3.8
Submitted
December 9, 2024
Published
2024-12-09

Abstract

A series of 5-aminoquinoline derivatives 3a-f and 3-aminophenol derivatives 5a-f were synthesized in order to determine their in vitro antimicrobial activity. The chemical structures of the synthesized compounds were confirmed by FT-IR and 1H NMR spectral studies. Among the synthesized compounds, 3a, 3e, 3f, 5b, 5c and 5f showed good antimicrobial activity against tested microbial strains.

References

  1. [1] Cimerman, Z.; Miljanic, S.; Galic, N. Croatica Chemica Acta 2000, 73, 81.
  2. [2] Singh, P.; Goel, R. L.; Singh, B. P. J. Indian Chem. Soc. 1975, 52, 958.
  3. [3] Perry, B. F.; Beezer, A. E.; Miles, R. J.; Smith, B. W.; Miller, J.; Nascimento, M. G. Microbois. 1988, 45, 181.
  4. [4] Elmali, A.; Kabak, M.; Elerman, Y. J. Mol. Struct. 2000, 477, 151.
  5. [5] Patel, P. R.; Thaker, B. T.; Zele, S. Indian J. Chem. 1999, 38, 563.
  6. [6] Patai, S. J. Wiley & Sons, London, 1970.
  7. [7] Jungreis, E.; Thabet, S. Marcell Dekker, New York, 1969.
  8. [8] Gawad, M. A.; Issa, Y. M.; Abd-Alhamid, S. M. Egypt J. Pharm. Sci. 1996, 73, 55.
  9. [9] Sari, N.; Arslan, S.; Logoglu, E.; Sariyan, I. G. U. J. Sci. 2003, 16, 283.
  10. [10] Opletalova, V.; Hartl, J.; Patel, A.; Palat, A.; Buchta, V. Farmaco 2002, 57, 135.
  11. [11] Biava, M.; Fioravanti, R.; Porretta, G. C.; Sleite, G.; Deidda, D.; Lampis, G.; Pompei, R. Farmaco 2002, 54, 721.
  12. [12] Ernest, H. GB 2078212, 1982.
  13. [13] Holla, B. S.; Rao, B. S.; Shridhara, K.; Akberali, P. M. Farmaco 2000, 55, 338.
  14. [14] Chaha, V. K.; Ranwa, N. S.; Dadheech, P. K. J. Phytol. Res. 1998, 11, 201.
  15. [15] Mehta, B. H.; Vengarlekar, V. P. Asian J. Chem. 1999, 11, 397.
  16. [16] Raman, N.; Muthuraj, V.; Ravichandran, S.; Kulandaisamy, A. Proc. Indian Acad. Sci. 2003, 115, 161.
  17. [17] Capdeville, R.; Buchdunger, E.; Zimmermann, J.; Matter,A. Nat. Rev. Drug. Discov. 2002, 1, 493.
  18. [18] Ignatovich, Z. V.; Kadutskii, A. P.; Koroleva, E. V.; Baranovskii, A. V.; Gusak, K. N. Russian Journal of Organic Chemistry 2009, 45, 1070.
  19. [19] Dubey, R. K.; Dubey, U. K.; Mishra, C. M. Indian Journal of Chemistry 2008, 47A, 1208.
  20. [20] Demir, I.; Bayrakcr, M.; MutluCimerman, Z.; Miljanic, S.; Galic, N. Croatica Chemica Acta 2000, 73, 81.
  21. [21] Singh, P.; Goel, R. L.; Singh, B. P. J. Indian Chem. Soc. 1975, 52, 958.
  22. [22] Perry, B. F.; Beezer, A. E.; Miles, R. J.; Smith, B. W.; Miller, J.; Nascimento, M. G. Microbois. 1988, 45, 181.
  23. [23] Elmali, A.; Kabak, M.; Elerman, Y. J. Mol. Struct. 2000, 477, 151.
  24. [24] Patel, P. R.; Thaker, B. T.; Zele, S. Indian J. Chem. 1999, 38, 563.
  25. [25] Patai, S. J. Wiley & Sons, London, 1970.
  26. [26] Jungreis, E.; Thabet, S. Marcell Dekker, New York, 1969.
  27. [27] Gawad, M. A.; Issa, Y. M.; Abd-Alhamid, S. M. Egypt J. Pharm. Sci. 1996, 73, 55.
  28. [28] Sari, N.; Arslan, S.; Logoglu, E.; Sariyan, I. G. U. J. Sci. 2003, 16, 283.
  29. [29] Opletalova, V.; Hartl, J.; Patel, A.; Palat, A.; Buchta, V. Farmaco 2002, 57, 135., K.; Pekacar, A. I. Acta Chim. Slov. 2008, 55, 120.
  30. [30] Ha, S. T.; Ong, L. K.; Win, Y. F.; Yeap, G. Y.; Bonde, N. L.; Boey, P. L. American Journal of Applied Sciences 2010, 7, 656-660.
  31. [31] Santosh, K.; Niranjan, M. S.; Chaluvaraju, K. C.; Jamakhandi, C. M.; Dayanand, K. Journal of Current Pharmaceutical Research 2010, 1, 39.
  32. [32] Roman, I. G.; Andree, M. Bulletin of the Chemists and Technologists of Macedonia 2001, 20, 131.
  33. [33] Bauer, A. W.; Kirby, W. M.; Sherris, J. C.; Turck, M. Am. J. Clin. Pathol. 1966, 45, 493.
  34. [34] Satish, S.; Mohana, D. C.; Raghavendra, M. P.; Raveesha, K. A. J. Agri. Techn. 2007, 3, 109.

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